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Product Name: GSK126 | EZH2 inhibitor
Product Description: GSK126 is an indole-based inhibitor of EZH2 methyltransferase activity, with an Ki-app of 0.5-3 nM independent of substrate used. It is competitive with S-adenosyl methionine (SAM) and non-competitive with peptide substrates. GSK126 is highly selective agWeb Site:Medchemexpress
Chemical Formula: C31H38N6O2
Molecular Weight: 526.67
‘&“CAS NO: 1449277-10-4 GNE-495
Purity: 99%
Appearance: White
Chemical Name: (S)-1-(sec-butyl)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamideAurora Kinase inhibitors
Solubility: Up to 50 mM in DMSO
Shipping Condition: The product is shipped in a glass vial at ambient temperature.
Storage Condition: For longer shelf life, store solid powder at 4oC desiccated, or store DMSO solution at -20oC.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/19773430

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Author: DNA_ Alkylatingdna