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Product Name: GSK6853
Chemical Name: (R)-N-(1,3-dimethyl-6-(2-methylpiperazin-1-yl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methoxybenzamide
SMILES Code: O=C(NC1=C(N2[[email protected]](C)CNCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
CAS NO: 1202055-32-0 Product: JZL 184
Synonym: GSK-6853; GSK 6853
Chemical Formula: C22H27N5O3Molecular Weight: 409.49
Appearance: Solid powderWeb Site:Medchemexpress
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Drug-Linker Conjugates for ADC inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/10381057

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Author: DNA_ Alkylatingdna