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Product Name: I-CBP 112
Chemical Name: (S)-1-(7-(3,4-dimethoxyphenyl)-9-((1-methylpiperidin-3-yl)methoxy)-2,3-dihydrobenzo[f][1,4]oxazepin-4(5H)-yl)propan-1-one
SMILES Code: CCC(N1CCOC2=C(OC[C@@H]3CN(C)CCC3)C=C(C4=CC=C(OC)C(OC)=C4)C=C2C1)=O
CAS NO: 1002789-86-7 Product: (±)-BI-D
Synonym: I-CBP112; I-CBP-112
Chemical Formula: C27H36N2O5Molecular Weight: 468.594
Appearance: Solid powderMedchemexpress
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).TAK1 inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: I-CBP112 is a selective inhibitor of the bromodomain-containing transcription factors CREBBP (CBP) and EP300 (IC50 = 0.142 and 0.625 μM, respectively). I-CBP112 has little activity against other bromodomains at concentrations up to 1 mM. I-CBP112 targets PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/19197797

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Author: DNA_ Alkylatingdna