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Product Name: MK-0974
Chemical Name: N-((3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-trifluoroethyl)azepan-3-yl)-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide
SMILES Code: O=C(N1CCC(N(C2=CC=CN=C2N3)C3=O)CC1)N[C@H]4C(N(CC(F)(F)F)C[C@H](C5=CC=CC(F)=C5F)CC4)=O
CAS NO: 141286-78-4 Product: Yunaconitine
Synonym: Telcagepant; MK0974; MK 0974
Chemical Formula: C26H27F5N6O3Molecular Weight: 566.533
Appearance: Solid powderWeb Site click
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Potassium Channel inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: MK-0974(Telcagepant) is a highly potent, selective, and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22037406

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Author: DNA_ Alkylatingdna