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Product Name: NVS-PAK1-1
Chemical Name: (S)-3-(2-Chloro-5-(2,2-difluoroethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-ylamino)-N-isopropylpyrrolidine-1-carboxamideTheoretical AnalysisMetonChem Cat#: MC7043012
SMILES Code:
CAS NO: 321-55-1 Product: Eprinomectin
Synonym:
Chemical Formula: C23H25ClF3N5OMolecular Weight: 479.93
Appearance: Solid powderMedchemexpress.com
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).HSP inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: NVS-PAK1-1 is a potent allosteric inhibitor of p21-activated kinase PAK1, a serine-threonine kinase that is upregulated in many cancers. NVS-PAK1-1 has an IC50 value of 5 nM for dephoshorylated PAK1 and 6 nM for phosphorylated PAK1 in an in vitro dephosphPubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22972527

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Author: DNA_ Alkylatingdna