Share this post on:

Product Name: OTX015
Chemical Name: (S)-2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide
SMILES Code: O=C(NC1=CC=C(O)C=C1)C[[email protected]]2C3=NN=C(C)N3C4=C(C(C)=C(C)S4)C(C5=CC=C(Cl)C=C5)=N2
CAS NO: 66108-95-0 Product: AMD 3465
Synonym: OTX-015; OTX 015; MK-8628; MK 8628; MK8628
Chemical Formula: C25H22ClN5O2SMolecular Weight: 491.992
Appearance: Solid powderWeb Site:Medchemexpress
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).URAT1 inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: OTX015 is a potent BET bromodomian inhibitor, which targets the BET bromodomain proteins 2, 3, and 4. It is the first BRD2/3/4 inhibitor to enter clinical trials.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/21239112

Share this post on:

Author: DNA_ Alkylatingdna