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Product Name: TC-G-1008
Chemical Name: N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide
SMILES Code: CS(=O)(NC1=CC=C(CNC2=NC(NC)=NC(C3=NC=CC=C3)=C2)C(Cl)=C1)=O
CAS NO: 849214-04-6 Product: Wilforine
Synonym: TC-G1008; TC-G 1008; TCG-1008; TCG1008; TCG 1008; GPR39-C3; GPR39C3; GPR39 C3
Chemical Formula: C18H19ClN6O2SMolecular Weight: 418.9
Appearance: Solid powderWeb Site:Medchemexpress
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).ADC Cytotoxin inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: TC-G-1008 (GPR39-C3) is potent and selective GPR39 agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively). TC-G-1008 is selective over a panel of kinases and displays minimal binding affinity for ghrelin and neurotensin-1 receptPubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/15839304

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Author: DNA_ Alkylatingdna