Product Name :
Orelabrutinib
Synonym :
Chemical Name :
CAS NO.:
1655504-04-3
Molecular formula :
C26H25N3O3
Molecular Weight:
427.5 g/mol
Classification :
MedChemExpress Products > Life Sciences > Ligands > Orelabrutinib
Description:
Orelabrutinib is a potent inhibitor of Bruton’s tyrosine kinase (BTK). It has been shown to inhibit the BTK enzyme in both human and mouse cells, which prevents activation of the B-cell receptor and inhibits immunoglobulin production. Orelabrutinib is also a 5-HT1A agonist and has been shown to have anti-cancer effects on drug-resistant acute lymphocytic leukemia. The drug binds to the active site of BTK as a covalent inhibitor, resulting in its inhibition. Orelabrutinib also acts as an antagonist at serotonin receptors 5-HT1A, leading to its potential therapeutic effects in autoimmune diseases.
Purity :
>98%
Specifications :
10 mM * 1 mL
Price.:
275
Price unit :
$
Inventory :
In stock
Related websites: https://www.medchemexpress.com
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