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Product Name: GSK126
Chemical Name: (S)-1-(sec-butyl)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide
SMILES Code: O=C(C1=CC(C2=CC=C(N3CCNCC3)N=C2)=CC4=C1C(C)=CN4[C@@H](C)CC)NCC5=C(C)C=C(C)NC5=O
CAS NO: 924296-17-3 Product: Taltirelin
Synonym: GSK-126; GSK 126
Chemical Formula: C31H38N6O2Molecular Weight: 526.67
Appearance: Solid powderWeb Site click
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Raf inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: GSK126 is a potent, highly selective, S-adenosyl-methionine-competitive, small-molecule inhibitor of EZH2 methyltransferase activity, which decreases global H3K27me3 levels and reactivates silenced PRC2 target genes.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/7828988

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Author: DNA_ Alkylatingdna