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Product Name: RQ-00203078
Chemical Name: 4-(N-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-(trifluoromethoxy)benzyl)sulfamoyl)benzoic acid
SMILES Code: O=C(O)C1=CC=C(S(=O)(N(C2=NC=C(C(F)(F)F)C=C2Cl)CC3=CC=C(OC(F)(F)F)C=C3)=O)C=C1
CAS NO: 1419949-20-4 Product: Indinavir (sulfate)
Synonym: RQ 00203078; RQ00203078
Chemical Formula: C21H13ClF6N2O5SMolecular Weight: 554.84
Appearance: Solid powderWeb Site click
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Mps1 inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: RQ-00203078 is a potent, selective and orally active TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively). RQ-00203078 blocks TRPM8 activity and reduces the invasion potential of oral squamous carcinoma cell lines. RQ-PubMed ID:http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2938305/

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Author: DNA_ Alkylatingdna